On drug discovery against infectious diseases and academic medicinal chemistry contributions

• Yves L. Janin

Beilstein J. Org. Chem. 2022, 18, 1355–1378, doi:10.3762/bjoc.18.141

• review [62] focusing on hit selection (triage) is probably a good general starting point to describe the problem which academics are facing: “It is increasingly clear that academic high-throughput screening (HTS) and virtual HTS triage suffers from a lack of scientists trained in the art and science of

Iridium-catalyzed hydroacylation reactions of C1-substituted oxabenzonorbornadienes with salicylaldehyde: an experimental and computational study

• Angel Ho,
• Austin Pounder,
• Krish Valluru,
• Leanne D. Chen and
• William Tam

Beilstein J. Org. Chem. 2022, 18, 251–261, doi:10.3762/bjoc.18.30

• the art and science of selective molecular engineering [1]. To date, organic synthesis has largely been governed by the interconversion of pre-existing functional groups through the use of more traditional transition-metal-catalyzed cross-coupling reactions [2][3][4][5]. Although these reactions have

Perspective isomorphs – a new classification of molecular structures based on artistic and chemical concepts

• Jannis Neumann,
• Ansgar Schnurr and
• Hermann A. Wegner

Beilstein J. Org. Chem. 2019, 15, 2319–2326, doi:10.3762/bjoc.15.224

• isomorphs and its discussions herein will extend current models and stimulate the discourse about the nature of atoms and molecules and especially their models. Keywords: art and science; nomenclature; perspective; representation in chemistry; structure; Introduction Up to now, epistemological concepts of

Organocatalysis

• Benjamin List

Beilstein J. Org. Chem. 2012, 8, 1358–1359, doi:10.3762/bjoc.8.156

• Benjamin List Max-Planck-Institut für Kohlenforschung, Kaiser-Wilhelm-Platz 1, D-45470 Mülheim an der Ruhr, Germany 10.3762/bjoc.8.156 Keywords: organocatalysis; During the past 12 years or so, hardly any other field has impacted the art and science of chemical synthesis more profoundly than

Functionalization of anthracene: A selective route to brominated 1,4-anthraquinones

• Kiymet Berkil Akar,
• Osman Cakmak,
• Orhan Büyükgüngör and
• Ertan Sahin

Beilstein J. Org. Chem. 2011, 7, 1036–1045, doi:10.3762/bjoc.7.118

• Kiymet Berkil Akar Osman Cakmak Orhan Buyukgungor Ertan Sahin Department of Chemistry, Faculty of Art and Science, Gaziosmanpasa University, 60250, Tokat, Turkey Department of Physics, Faculty of Art and Science, Ondokuzmayıs University, 55060, Samsun, Turkey Department of Chemistry, Faculty of

• Art and Science, Atatürk University, 25240, Erzurum, Turkey 10.3762/bjoc.7.118 Abstract Efficient and stereoselective syntheses are described for the preparation of 2,3,9,10-tetrabromo-1,4-dimethoxy-1,2,3,4-tetrahydroanthracenes 7, 8 and the corresponding 1,4-diol 17 by silver ion-assisted solvolysis

Highly brominated anthracenes as precursors for the convenient synthesis of 2,9,10-trisubstituted anthracene derivatives

• Osman Cakmak,
• Leyla Aydogan,
• Kiymet Berkil,
• Ilhami Gulcin and
• Orhan Buyukgungor

Beilstein J. Org. Chem. 2008, 4, No. 50, doi:10.3762/bjoc.4.50

• Osman Cakmak Leyla Aydogan Kiymet Berkil Ilhami Gulcin Orhan Buyukgungor Gaziosmanpasa University, Faculty of Art and Science, Department of Chemistry, TR-60240, Tokat, Turkey Ataturk University, Faculty of Art and Science, Department of Chemistry, TR-25240, Erzurum, Turkey Ondokuzmayis University

• , Faculty of Art and Science, Department of Physics, TR-55060, Samsun, Turkey (author to whom inquries concerning the X-ray structure should be directed) 10.3762/bjoc.4.50 Abstract When 9,10-dibromoanthracene was treated with bromine in CCl4 without a catalyst, 1,2,3,4,9,10-hexabromo-1,2,3,4